Fmoc-L-Pro(4-guanidino-Pbf)-OH (2S,4R)

Chemical name: (2S,4R)-1-(9-Fluorenylmethyloxycarbonyl)-4-(3-(2,2,4,6,7-pentamethyl-2,3-dihydrobenzofuran-5-ylsulfonyl)guanidino)pyrrolidine-2-carboxylic acid // Synonyms: (2S,4R)-Fmoc-4-(N'-Pbf-guanidino)-pyrrolidine-2-carboxylic acid,(2S,4R)-1-(((9H-fluoren-9-yl)methoxy)carbonyl)-4-(3-(2,2,4,6,7-pentamethyl-2,3-dihydrobenzofuran-5-ylsulfonyl)guanidino)pyrrolidine-2- carboxylic acid, Fmoc-Pro(4-guanidino-Pbf)-OH(2S,4

  • Product code:FAA5220
  • CAS No.:1864002-98-1
  • Formula:C34H38N4O7S
  • Molecular weight:646.75 g/mol

Starting at $390.00

Grouped product items
Qty Packing unit Price SKU
250 mg
1 g

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Plasmid DNA delivery by arginine-rich cell-penetrating peptides containing unnatural amino acids; T. Kato, H. Yamashita, T. Misawa, K. Nishida, M. Kurihara, M. Tanaka, Y. Demizu, M. Oba; Bioorg. Med. Chem. 2016; 24(12): 2681-2687.

Substitution of Arginine with Proline and Proline Derivatives in Melanocyte-Stimulating Hormones Leads to Selectivity for Human Melanocortin 4 Receptor; H. Qu, M. Cai, A. V. Mayorov, P. Grieco, M. Zingsheim, D. Trivedi, V. J. Hruby; J. Med. Chem. 2009; 52(12): 3627-3635.

Rational Design of a-Conotoxin Analogues Targeting a7 Nicotinic Acetylcholine Receptors; C. Armishaw, A. A. Jensen, T. Balle, R. J. Clark, K. Harpsøe, C. Skonberg, T. Liljefors, K. Strømgaard; J. Biol. Chem. 2009; 284(14): 9498-9512.

Synthesis of Proteins Containing Modified Arginine Residues; A. K. Choudhury, S. Y. Golovine, L. M. Dedkova, S. M. Hecht; Biochem. 2007; 46(13): 406-4076.

Practical and Efficient Synthesis of Orthogonally Protected Constrained 4-Guanidinoprolines; M. Tamaki, G. Han, V. J. Hruby; J. Org. Chem. 2001; 66(3): 1038-1042.

Synthesis of Alanine and Proline Amino Acids with Amino or Guanidinium Substitution on the Side Chain; Z. Zhang, A. V. Aerschot, C. Hendrix, R. Busson, F. David, P. Sandra, P. Herdewijn; Tetrahedron 2000; 56(16): 2513-2522.

Conformationally restricted arginine analogs; T. R. Webb, C. Eigenbrot; J. Org. Chem. 1991; 56(9): 3009-3016.

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